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Olodaterol hydrochloride

CAS No. 869477-96-3

Olodaterol hydrochloride ( BI1744 CL )

产品货号. M16316 CAS No. 869477-96-3

Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥640 有现货
5MG ¥988 有现货
10MG ¥1604 有现货
25MG ¥2989 有现货
50MG ¥4447 有现货
100MG ¥6383 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Olodaterol hydrochloride
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
  • 产品描述
    Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2; shows >250 fold selectivity over hβ1; exerts a bronchodilatory efficacy over 24 h in dogs and guinea pigs in the absence of systemic pharmacodynamic effects.COPD Phase 3 Clinical
  • 同义词
    BI1744 CL
  • 通路
    Angiogenesis
  • 靶点
    Adrenergic Receptor
  • 受体
    hβ2-adrenoceptor
  • 研究领域
    Inflammation/Immunology
  • 适应症
    COPD

化学信息

  • CAS Number
    869477-96-3
  • 分子量
    413.90
  • 分子式
    C21H17ClFN3OS
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: 50 mg/mL; Water: 15 mg/mL ( < 1 mg/ml refers to the product slightly soluble or insoluble )
  • SMILES
    CC(C)(CC1=CC=C(C=C1)OC)NCC(C2=C3C(=CC(=C2)O)NC(=O)CO3)O.Cl
  • 化学全称
    4-(4-(4-fluorophenyl)-2-(4-(methylsulfinyl)phenyl)-1H-imidazol-5-yl)pyridine hydrochloride

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Bouyssou T, et al. Bioorg Med Chem Lett. 2010 Feb 15;20(4):1410-4.
2. Bouyssou T, et al. J Pharmacol Exp Ther. 2010 Jul;334(1):53-62.
3. Wex E, et al. Br J Pharmacol. 2015 Jul;172(14):3537-47.
产品手册
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