Olodaterol hydrochloride
CAS No. 869477-96-3
Olodaterol hydrochloride ( BI1744 CL )
产品货号. M16316 CAS No. 869477-96-3
Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥640 | 有现货 |
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5MG | ¥988 | 有现货 |
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10MG | ¥1604 | 有现货 |
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25MG | ¥2989 | 有现货 |
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50MG | ¥4447 | 有现货 |
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100MG | ¥6383 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Olodaterol hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
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产品描述Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2; shows >250 fold selectivity over hβ1; exerts a bronchodilatory efficacy over 24 h in dogs and guinea pigs in the absence of systemic pharmacodynamic effects.COPD Phase 3 Clinical
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同义词BI1744 CL
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通路Angiogenesis
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靶点Adrenergic Receptor
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受体hβ2-adrenoceptor
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研究领域Inflammation/Immunology
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适应症COPD
化学信息
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CAS Number869477-96-3
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分子量413.90
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分子式C21H17ClFN3OS
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纯度>98% (HPLC)
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溶解度DMSO: 50 mg/mL; Water: 15 mg/mL ( < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESCC(C)(CC1=CC=C(C=C1)OC)NCC(C2=C3C(=CC(=C2)O)NC(=O)CO3)O.Cl
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化学全称4-(4-(4-fluorophenyl)-2-(4-(methylsulfinyl)phenyl)-1H-imidazol-5-yl)pyridine hydrochloride
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Bouyssou T, et al. Bioorg Med Chem Lett. 2010 Feb 15;20(4):1410-4.
2. Bouyssou T, et al. J Pharmacol Exp Ther. 2010 Jul;334(1):53-62.
3. Wex E, et al. Br J Pharmacol. 2015 Jul;172(14):3537-47.
2. Bouyssou T, et al. J Pharmacol Exp Ther. 2010 Jul;334(1):53-62.
3. Wex E, et al. Br J Pharmacol. 2015 Jul;172(14):3537-47.
产品手册
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